GSK-2807 free base
Product Specifications
CAS Number
2245255-65-4
Target
Histone Methyltransferase, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
GSK2807 is a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM) . GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 may be useful for cancer treatment.
Smiles
O[C@H]1[C@H](N2C=3C(N=C2)=C(N)N=CN3)O[C@H](CN(CC[C@@H](C(O)=O)N)CCCN(C)C)[C@H]1O
Molecular Formula
C19H32N8O5
Molecular Weight
452.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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