TG11-77 free base
Product Specifications
CAS Number
2490544-33-5
Target
Others
Related Pathways
Others
Bioactivity
TG11-77 free base is a novel, Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist. TG11-77 free base has a Schild KB of 9.7 nM on EP2, a water solubility of 2.5 mM, a brain-to-plasma ratio of 0.4, and a plasma half-life of 2.4 h in mice. TG11-77 free base are representative second generation EP2 antagonists with improved pharmacodynamic and pharmacokinetic properties.
Smiles
C(CNC(=O)C=1C=NC(NC2=CC(C)=CC(C)=N2)=NC1)C=3C=4C(NC3C)=CC=CC4
Molecular Formula
C23H24N6O
Molecular Weight
400.48
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
MBS1376532-01 0.02 mg (E-Coli)
Recombinant Deinococcus geothermalis DNA replication and repair protein recF (recF)
Ask
View Details