SRX3212
Product Specifications
CAS Number
2735720-80-4
Target
Others
Related Pathways
Others
Bioactivity
SRX3212 is a Novel BRD4/PI3Kα inhibitor, displaying an IC50 of 3.7 nM toward BRD4BD1 and 32 nM toward BRD4BD2, and therefore was~65-fold more potent inhibitor of BRD4BD1 and~48-fold more potent inhibitor of BRD4BD2 than SF2523 (GLXC-10641), retaining its high inhibitory activity for PI3Kα (IC50: 22 nM) .
Smiles
O=C1C2=C(C(=CS2)C3=CC(C(NCC=4C=CC=NC4)=O)=C5C(=C3)OCCO5)OC(=C1)N6CCOCC6
Molecular Formula
C26H23N3O6S
Molecular Weight
505.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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