What is the catalog number for YM-202074?

The catalog number for YM-202074 is T69489.

What sizes are available for YM-202074?

YM-202074 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does YM-202074 come in?

YM-202074 is available in 3 different pack sizes.

Is YM-202074 in stock?

YM-202074 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures YM-202074?

YM-202074 is manufactured by Molfinity.

What is the estimated delivery time for YM-202074?

Estimated delivery time for YM-202074 is approximately 10 business day(s), depending on your location.

YM-202074

Product Specifications

CAS Number

299900-83-7

Target

Others, GluR

Related Pathways

Others, Neuroscience

Bioactivity

YM-202074 is a high affinity, selective metabotropic glutamate receptor type 1 (mGlu1) antagonist. YM-202074 binds an allosteric site of the rat mGlu1 receptor with a Ki of 4.8 nM. It inhibits mGlu1-mediated inositol phosphates production (IC50 = 8.6 nM in rat cerebellar granule cells) .