Vestipitant
Product Specifications
CAS Number
334476-46-9
Target
Others, Neurokinin receptor
Related Pathways
Neuroscience, GPCR/G Protein, Others
Bioactivity
Vestipitant, also known as GW597599, is one of the most potent and selective NK (1) receptor antagonists ever discovered, showing appropriate pharmacokinetic properties and in vivo activity. Its actions support the utility of NK (1) receptor blockade in the alleviation of anxiety and, possibly, depression. It is under development as a potential antiemetic and anxiolytic drug, and as a treatment for tinnitusand insomnia.
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C(N([C@H](C)C1=CC(C(F)(F)F)=CC(C(F)(F)F)=C1)C)(=O)N2[C@H](CNCC2)C3=C(C)C=C(F)C=C3
Molecular Formula
C23H24F7N3O
Molecular Weight
491.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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