What is the catalog number for SKF89976A HCl?

The catalog number for SKF89976A HCl is T68550.

What sizes are available for SKF89976A HCl?

SKF89976A HCl is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does SKF89976A HCl come in?

SKF89976A HCl is available in 3 different pack sizes.

Is SKF89976A HCl in stock?

SKF89976A HCl is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures SKF89976A HCl?

SKF89976A HCl is manufactured by Molfinity.

What is the estimated delivery time for SKF89976A HCl?

Estimated delivery time for SKF89976A HCl is approximately 10 business day(s), depending on your location.

SKF89976A HCl

Product Specifications

CAS Number

85375-85-5

Target

GABA Receptor, Others

Related Pathways

Neuroscience, Others, Membrane transporter/Ion channel

Bioactivity

SKF89976A is a potent GABA uptake inhibitor, which is selective for GAT-1 (IC50 values are 0.13, 550, 944 and 7210 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively) . SKF89976A inhibits transport current competitively (Ki = 7 μM) and transmitter-gated current non-competitively (Ki = 0.03 nM) . It is able to pass the blood-brain barrier after systemic administration and is active in vivo.