Cerlapirdine hydrochloride
Product Specifications
CAS Number
925447-04-7
Target
5-HT Receptor, Others
Related Pathways
GPCR/G Protein, Others, Neuroscience
Bioactivity
Cerlapirdine, also known as SAM-531, WAY-262,531 and PF-05212365, is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine has been in clinical development for the treatment of cognitive disorders associated with Alzheimer's disease and schizophrenia. As of 2011, it is in phase II clinical trials, and has demonstrated a trend toward efficacy along with a good side effect profile and no incidence of serious adverse events. It exerts its effects by acting as a selective 5-HT6 receptor antagonist.
Smiles
Cl.CN(C)CCCOc1ccc2[nH]nc(c2c1)S(=O)(=O)c1cccc2ccccc12
Molecular Formula
C22H24ClN3O3S
Molecular Weight
445.96
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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