Saterinone
Product Specifications
CAS Number
102669-89-6
Target
PDE, Adrenergic Receptor
Related Pathways
Neuroscience, GPCR/G Protein, Metabolism
Purity
>99.99%
Bioactivity
Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3 x 10 (-5) mol/l.
Smiles
CC1=C(C=C(C#N)C(=O)N1)C2=CC=C(OCC(CN3CCN(CC3)C4=C(OC)C=CC=C4)O)C=C2
Molecular Formula
C27H30N4O4
Molecular Weight
474.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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