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PARP10-IN-3

Product Specifications

CAS Number

2225800-19-9

Target

PARP

Related Pathways

DNA Damage/DNA Repair, Chromatin/Epigenetic

Purity

0.9954

Bioactivity

PARP10-IN-3 is a potent and selective mono-Adp-ribotransferase PARP10 inhibitor that inhibits human PARP10 (IC50:480 nM) . PARP10-IN-3 also inhibited human PARP2 and human PARP15 with IC50 values of 1.7 μM.

Smiles

O(C1=CC(C(N)=O)=CC=C1)C2=CC=C(C(N)=O)C=C2

Molecular Formula

C14H12N2O3

Molecular Weight

256.26

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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