What is the catalog number for GRP78-IN-3?

The catalog number for GRP78-IN-3 is T67897.

What sizes are available for GRP78-IN-3?

GRP78-IN-3 is available in the following size(s): 1 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 500 mg.

How many pack sizes does GRP78-IN-3 come in?

GRP78-IN-3 is available in 7 different pack sizes.

Is GRP78-IN-3 in stock?

GRP78-IN-3 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GRP78-IN-3?

GRP78-IN-3 is manufactured by Molfinity.

What is the estimated delivery time for GRP78-IN-3?

Estimated delivery time for GRP78-IN-3 is approximately 10 business day(s), depending on your location.

GRP78-IN-3

Product Specifications

CAS Number

2707510-30-1

Target

HSP

Related Pathways

Metabolism, Cytoskeletal Signaling

Purity

0.9949

Bioactivity

GRP78-IN-3, a potent small-molecule-competitive inhibitor of Hsp70 substrate binding and is a selective Grp78 (HSPA5) inhibitor with an IC50 of 0.59 μM. GRP78-IN-3 is 7-fold selective for HspA5 compared to HspA9 (IC50 of 4.3 μM) and >20-fold selective for HspA5 compared to HspA2 (IC50 of 13.9 μM) .