BJJF078
Product Specifications
CAS Number
2531244-56-9
Target
Glutaminase
Related Pathways
Proteases/Proteasome
Purity
0.9956
Bioactivity
BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.BJJF078 inhibits TG1 enzyme, with an IC50 of 0.16 μM.BJJF078 can be used to study multiple sclerosis (MS) . BJJF078 can be used to study multiple sclerosis (MS) .
Smiles
S(=O)(=O)(C=1C2=C(C(NC(=O)C3=CC(OC)=C(OC)C=C3)=CC=C2)C=CC1)N4CCC(NC(C=C)=O)CC4
Molecular Formula
C27H29N3O6S
Molecular Weight
523.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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