MCT1-IN-3
Product Specifications
CAS Number
2878360-80-4
Target
P-gp, Monocarboxylate transporter
Related Pathways
Membrane transporter/Ion channel, Neuroscience
Purity
0.9935
Bioactivity
MCT1-IN-3 is a monocarboxylate transporter 1 (MCT1) inhibitor, targeting solute carrier (SLC) monocarboxylate transporter 1 (MCT1; SLC16A1) for cancer treatment. MCT1-IN-3 (compound 24) showed the highest MCT1 transport inhibition with an IC50 value of 81.0 Nm and also exhibits significant inhibitory activity against the multidrug transporter ABCB1.
Smiles
C(=C(C(OC)=O)C#N)C=1C=2C(N(CC(NC3=CC=C(OC)C=C3)=O)C1)=CC=CC2
Molecular Formula
C22H19N3O4
Molecular Weight
389.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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