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H3R antagonist 7

Product Specifications

Target

Histamine Receptor

Related Pathways

GPCR/G Protein, Immunology/Inflammation, Neuroscience

Bioactivity

H3R antagonist 7 (compounds 4) is a histamine subtype 3 receptor (H3R) antagonist with a Ki value of 3.15 nM. It can potentially be used as a PET radioligand in the study of central nervous system (CNS) diseases.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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