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Enpp-1/3-IN-1

Product Specifications

Target

PDE|||CD73|||Phosphatase

Related Pathways

Immunology/Inflammation|||Metabolism

Bioactivity

Enpp-1/3-IN-1 (Compound 5j) serves as an inhibitor for ENPP1 and ENPP3, with IC50 values of 0.59 ?M for h-ENPP1 and 0.62 ?M for h-ENPP3, respectively. This compound also inhibits e5?NT (CD73) and TNAP, exhibiting IC50 values of 0.89 ?M for h-e5?NT, 5.12 ?M for r-e5?NT, and 1.68 ?M for h-TNAP. Enpp-1/3-IN-1 is applicable in cancer research.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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