What is the catalog number for DPP-4-IN-17?

The catalog number for DPP-4-IN-17 is T212193.

What sizes are available for DPP-4-IN-17?

DPP-4-IN-17 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does DPP-4-IN-17 come in?

DPP-4-IN-17 is available in 2 different pack sizes.

Is DPP-4-IN-17 in stock?

DPP-4-IN-17 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures DPP-4-IN-17?

DPP-4-IN-17 is manufactured by Molfinity.

What is the estimated delivery time for DPP-4-IN-17?

Estimated delivery time for DPP-4-IN-17 is approximately 10 business day(s), depending on your location.

DPP-4-IN-17

Product Specifications

Target

Proteasome

Related Pathways

Ubiquitination, Proteases/Proteasome

Bioactivity

DPP-4-IN-17 is an orally active and selective inhibitor of dipeptidyl peptidase-4 (DPP-4) with an IC50 value of 0.12 nM. It increases the enzyme's Km value (75.73 μM compared to the substrate alone at 27.18 μM) and reduces catalytic efficiency. In Streptozotocin (STZ) /Nicotinamide (NA) -induced diabetic rats, DPP-4-IN-17 lowers blood glucose levels and reverses weight loss. This compound is useful for research in type 2 diabetes (T2DM) .