Rel-A-395 hydrochloride
Product Specifications
CAS Number
2747996-65-0
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
Rel-A-395 hydrochloride is the relative configuration of A-395 hydrochloride. A-395 is an antagonist of protein-protein interactions within the polycomb repressive complex 2 (PRC2) . It inhibits the trimeric PRC2 complex (EZH2-EED-SUZ12) with an IC50 value of 18 nM.
Smiles
FC1=C2C(CCC2=CC=C1)N3C[C@@H]([C@@H](N(C)C)C3)C4=CC=C(C=C4)N5CCN(S(C)(=O)=O)CC5.Cl
Molecular Formula
C26H36ClFN4O2S
Molecular Weight
523.11
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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