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Sonvuterkib

Product Specifications

CAS Number

2890225-50-8

Target

ERK

Related Pathways

MAPK

Bioactivity

Sonvuterkib (WX001) is a potent and orally active inhibitor of extracellular signal-regulated kinases (ERK), exhibiting IC50 values of 1.4 nM for ERK1 and 0.54 nM for ERK2. It effectively inhibits cell proliferation and possesses anticancer properties.

Smiles

O=C1C=2N=C(SC2C3(N1CC4=NC(=CC=C4)C)COC3)C=5N=C(N=CC5C)NC6=CC=NN6C

Molecular Formula

C23H22N8O2S

Molecular Weight

474.54

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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