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PAD2/4-IN-1

Product Specifications

Target

PAD, Potassium Channel

Related Pathways

Membrane transporter/Ion channel, Chromatin/Epigenetic

Bioactivity

PAD2/4-IN-1 is an orally active inhibitor of PAD2 and PAD4, with IC50 values of 23 and 10 nM, respectively. It inhibits protein citrullination in neutrophils and reduces hERG channel toxicity. PAD2/4-IN-1 is applicable in research on autoimmune diseases, neurological disorders, and cancer.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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