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EZH2-IN-200

Product Specifications

CAS Number

1403257-80-6

Target

Histone Methyltransferase

Related Pathways

Chromatin/Epigenetic

Purity

0.9981

Bioactivity

EZH2-IN-200 (compound 30) is an effective EZH2 (Enhancer of Zeste homologue 2) inhibitor with an IC50 of 11 nM against EZH2, suitable for studying hematologic malignancies and solid tumors.

Smiles

O=C(NCC=1C(=O)NC(=CC1C)C)C2=CC(Br)=CC(=C2C)N(CC)C3CCOCC3

Molecular Formula

C23H30BrN3O3

Molecular Weight

476.41

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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