Anticancer agent 276
Product Specifications
Target
VEGFR, Estrogen Receptor/ERR, c-Met/HGFR, EGFR, Topoisomerase
Related Pathways
JAK/STAT signaling, Angiogenesis, DNA Damage/DNA Repair, Tyrosine Kinase/Adaptors, Endocrinology/Hormones
Bioactivity
Anticanceragent 276 (Compound 5) is a multitarget anticancer compound. It exhibits potent antitumor activity against human cancer cells, with IC50 values of 6.90 μM for HEPG2 cells and 4.48 μM for MCF7 cells. Anticanceragent 276 interacts strongly and stably with multiple targets, including topoisomerase II, VEGFR2, c-Met, EGFR, and ERα.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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