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PPARγ agonist 19

Product Specifications

Target

PPAR, COX

Related Pathways

Neuroscience, DNA Damage/DNA Repair, Immunology/Inflammation, Metabolism

Bioactivity

PPARγ agonist19 (Compound 5e) is a PPARγ agonist with an IC50 of 11.27 μM for COX-1 and 0.05 μM for COX-2. It enhances glucose uptake in rat hemidiaphragm assays more effectively than pioglitazone. Additionally, PPARγ agonist19 reduces hyperglycemia and insulin resistance in type 2 diabetic rat models and protects against renal and lipid damage caused by metabolic dysfunction.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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