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TK-684

Product Specifications

Target

Apoptosis, Phosphatase

Related Pathways

Apoptosis, Metabolism

Bioactivity

TK-684 is a potent and selective allosteric inhibitor of SHP2, with IC50 values of 2.1 nM for SHP2WT and greater than 1000 nM for SHP2PTP. It inhibits cell proliferation and induces apoptosis (apoptosis) . Additionally, TK-684 reduces the protein expression of p-AKT and p-ERK.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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