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MS115

Product Specifications

Target

Histone Methyltransferase, PROTACs

Related Pathways

Chromatin/Epigenetic, PROTAC

Bioactivity

MS115 is a selective PRMT5/MEP50 PROTAC degrader with DC50 values of 17.4 nM for PRMT5 and 11.3 nM for PRMT5 in MDAMB468 cells after 24 hours. MS115 also inhibits the proliferation of breast cancer cells.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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