CYP1B1-IN-9
Product Specifications
CAS Number
3077254-39-5
Target
Cytochromes P450
Related Pathways
Metabolism
Bioactivity
CYP1B1-IN-9 is a highly selective and competitive CYP1B1 inhibitor, with IC50 values of 1.48 nM for CYP1B1, and greater than 100 μM and 80 μM for CYP1A1 and CYP1A2, respectively. This compound effectively inhibits the migration and invasion of A549/T cells, offers the potential to resensitize paclitaxel-resistant cells, and exhibits good metabolic stability and safety, as well as favorable pharmacokinetic properties. CYP1B1-IN-9 is applicable in research on tumor resistance.
Smiles
O=C(NC=1C=C(Cl)C=C(Cl)C1)C2=NC(=CS2)C=3C=CC=C(Cl)C3
Molecular Formula
C16H9Cl3N2OS
Molecular Weight
383.68
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC041866-500 1x 500 µL
Calponin-1 (Smooth Muscle Marker) (rCNN1/832), CF405S conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
![ASS1 Mouse Monoclonal Antibody [Clone ID: OTI1B10]](https://cdn.genprice.uk/products/937/68dd18ba061270361e9084dd/imageurl/cf809119.webp)
