Antiproliferative agent-71

Product Specifications

CAS Number

3083307-42-7

Target

Androgen Receptor|||Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic|||Endocrinology/Hormones

Bioactivity

Antiproliferative agent-71 (Compound II-5) is an orally active dual inhibitor that targets both the androgen receptor (AR) and bromodomain-containing protein 4 (BRD4) . By inhibiting the functions of AR and BRD4 simultaneously, Antiproliferative agent-71 effectively suppresses the growth and proliferation of tumor cells. This compound holds potential for research in prostate cancer.

Smiles

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