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P2Y1 antagonist 2

Product Specifications

Target

P2Y Receptor

Related Pathways

GPCR/G Protein|||Neuroscience

Bioactivity

P2Y1 antagonist 2 (Compound 19) is a P2Y1 receptor antagonist with an IC50 of 0.49 ?M. It exhibits significant anti-platelet aggregation activity by inhibiting the P2Y1 receptor. Additionally, this compound elevates nuclear Nrf2 protein levels, showing neuroprotective effects against oxidative stress damage. P2Y1 antagonist 2 effectively reduces cerebral infarction size and improves neurological function, making it useful for ischemic stroke research.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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