AAK1-IN-8

Product Specifications

CAS Number

2969205-90-9

Target

Serine/threonin kinase|||AAK1 (AP2 associated kinase 1)

Related Pathways

Cell Cycle/Checkpoint|||Neuroscience|||Metabolism

Bioactivity

AAK1-IN-8 (Compound 18) is a broad-spectrum NAK inhibitor. It effectively inhibits AAK1 and GAK with EC50 values of 50 nM and 190 nM, respectively, and prevents the phosphorylation of the AP2-µ2 subunit at threonine 156 (T156) .

Smiles

O=C(NCC=1C=CC=CC1)C2=CC=C3C=C2OCCOCCN=C4C=CN5N=CC3=C5N4

Molecular Formula

C24H23N5O3

Molecular Weight

429.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

NBP3-06986AF647 0.1 mL

Rabbit Polyclonal p16INK4a/CDKN2A Antibody [Alexa Fluor 647]

Ask

View Details

abx682070-01 10 µg

Human Glutathione S-Transferase Omega 1 (GSTO1) Protein

Ask

View Details

abx682070-02 100 µg

Human Glutathione S-Transferase Omega 1 (GSTO1) Protein

Ask

View Details

abx682070-03 1 mg

Human Glutathione S-Transferase Omega 1 (GSTO1) Protein

Ask

View Details

E55A11215 100 µL

Human GOLM1/GP73 Monoclonal Antibody

Ask

View Details

E3565-17F 100 µg

Estrogen Receptor b1, b2, Rat (ERb1, 2) Control Peptide

Ask

View Details