ESC1002755
Product Specifications
CAS Number
2915567-21-2
Target
Dehydrogenase
Related Pathways
Metabolism
Bioactivity
ESC1002755 is an inhibitor of 17β-HSD10 with an IC50 of 19 nM. Notably enzyme-specific, ESC1002755 exhibits non-competitive inhibition against the cofactor NADH. At a concentration of 50 μM, it shows minimal cytotoxicity in HEK293 cells. It holds potential for research in Alzheimer's disease and hormone-dependent cancers such as prostate, bone, and colorectal cancers.
Smiles
C(=O)(N1[C@@H](CCC1)C2=C(C=CC=C2)C3=CC(O)=CC=C3)C=4SC=CC4Cl
Molecular Formula
C21H18ClNO2S
Molecular Weight
383.89
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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