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FLT3-IN-32

Product Specifications

CAS Number

3047195-48-9

Target

FLT|||Apoptosis

Related Pathways

Angiogenesis|||Apoptosis|||Tyrosine Kinase/Adaptors

Bioactivity

FLT3-IN-32 is a potent FLT3 inhibitor with high selectivity, effectively suppressing FLT3 activating mutations and inducing apoptosis. It demonstrates good tolerance in non-tumor-bearing mice. In NOD/SCID mice loaded with MV4-11 cells, FLT3-IN-32 exhibits outstanding antitumor efficacy, significantly extending mouse survival. FLT3-IN-32 is applicable for acute myeloid leukemia research.

Smiles

O=C(NC1=NOC(=C1)C(C)(C)C)NC=2C=CC=3OC(=CC3C2)C(=O)C4=CC=5C(=CC=C(O)C5CN(C)C)N4

Molecular Formula

C28H29N5O5

Molecular Weight

515.56

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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