ER degrader 11
Product Specifications
CAS Number
2770911-29-8
Target
Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Bioactivity
ER degrader 11 (Compound 5) is an orally active, brain-penetrant, and selective estrogen receptor degrader, with an ERα IC50 of 1.6 nM. It holds potential for research into breast cancer brain metastasis.
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C[C@H]1N(C23CC(C2)C3)[C@@H](C4=C(C1)C=5C(N4)=CC=CC5)C6=C(F)C=C(NC7CN(CCCF)C7)C=C6F
Molecular Formula
C29H33F3N4
Molecular Weight
494.59
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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