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Dyrk1A-IN-9

Product Specifications

Target

DYRK

Related Pathways

Cell Cycle/Checkpoint, Tyrosine Kinase/Adaptors

Bioactivity

Dyrk1A-IN-9 (Compound L9) is a moderately active DYRK1A inhibitor with an IC50 of 1.67 μM. It demonstrates neuroprotective activity by regulating Aβ expression and Tau protein phosphorylation. Dyrk1A-IN-9 is applicable for Alzheimer's disease research.

Molecular Formula

C11H10N8

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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