α2AR agonist 1
Product Specifications
Target
Adrenergic Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
α2AR agonist 1 (compound S6a) is a morpholinopyrimidinone that serves as an agonist for the α2-adrenergic receptor (α2AR) . This compound elicits a concentration-dependent relaxation in precontracted aortic rings induced by phenylephrine (pEC50=6.81) . Additionally, α2AR agonist 1 elevates levels of NOx and NO in HUVEC.
Molecular Formula
C16H15N4NaO2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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