Antitumor agent-180
Product Specifications
Target
Apoptosis
Related Pathways
Apoptosis
Bioactivity
Antitumor agent-180 (Compound 13a) is an inhibitor of BUB1 mitotic checkpoint serine/threonine kinase B (BUB1B) . It suppresses the proliferation of ccRCC cells Caki-1 with an IC50 of 2.047 μM and induces necrosis and apoptosis in Caki-1 cells.
Molecular Formula
C34H41N9O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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