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Antitumor agent-180

Product Specifications

Target

Apoptosis

Related Pathways

Apoptosis

Bioactivity

Antitumor agent-180 (Compound 13a) is an inhibitor of BUB1 mitotic checkpoint serine/threonine kinase B (BUB1B) . It suppresses the proliferation of ccRCC cells Caki-1 with an IC50 of 2.047 μM and induces necrosis and apoptosis in Caki-1 cells.

Molecular Formula

C34H41N9O

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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