CDD-2807
Product Specifications
Target
C-RET, Serine Protease, CDK
Related Pathways
Apoptosis, Tyrosine Kinase/Adaptors, Proteases/Proteasome, Cell Cycle/Checkpoint
Bioactivity
CDD-2807 is a serine/threonine kinase 33 (STK33) inhibitor with an IC50 of 9.2 nM. In mice, CDD-2807 demonstrates no significant toxicity and can cross the blood-testis barrier without accumulating in the brain. It offers reversible contraceptive effects, indicating potential for development as a male contraceptive.
Molecular Formula
C29H26N4O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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