CFTR potentiator 1
Product Specifications
Target
CFTR
Related Pathways
Membrane transporter/Ion channel
Bioactivity
CFTRpotentiator 1 (I1421) is a potent CFTR potentiator with an EC50 value of 64 nM. It allosterically activates various mutations causing cystic fibrosis, such as ΔF508 and G551DCFTR.
Molecular Formula
C18H18N4O3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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