VCC972839:01
Product Specifications
Target
Apoptosis, CDK
Related Pathways
Cell Cycle/Checkpoint, Apoptosis
Bioactivity
VCC972839:01 is an inhibitor of cyclin-dependent kinase (CDK9) with an IC50 value of 7 nM. It inhibits the viability of SCLC cells at nanomolar concentrations and induces apoptosis through the intrinsic pathway. Additionally, VCC972839:01 demonstrates antitumor activity in mouse models.
Molecular Formula
C24H20N6O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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