Thailanstatin A cyclohexane diamine formic
Product Specifications
Target
Drug-Linker Conjugates for ADC
Related Pathways
Antibody-drug Conjugate/ADC Related
Bioactivity
Thailanstatin A cyclohexane diamine formic is an analogue of Spliceostatin. It effectively inhibits the proliferation of various cells, including N87 (IC50 = 0.33 ?M), BT474 (IC50 = 0.34 ?M), MDA-MB-361-DYT2 (IC50 = 0.88 ?M), and MDA-MB-468 (IC50 = 0.27 ?M) . Additionally, Thailanstatin A cyclohexane diamine formic can be utilized as a drug-linker conjugate in ADC (antibody-drug conjugate) molecules.
Molecular Formula
C35H55N3O10
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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