HCYP1B1-IN-2
Product Specifications
CAS Number
3043683-33-3
Target
Cytochromes P450, Aryl Hydrocarbon Receptor
Related Pathways
Immunology/Inflammation, Metabolism
Bioactivity
HCYP1B1-IN-2 (compound 3n) is a potent inhibitor of the human enzyme cytochrome P450 1B1 (hCYP1B1) . It exhibits strong anti-hCYP1B1 activity with an IC50 of 0.040 nM and can also block AhR transcriptional activity. hCYP1B1-IN-2 effectively inhibits hCYP1B1 through a mixed inhibition mode with a Ki value of 21.71 pM.
Smiles
O=C1C=2C=CC=C3C(Br)=CC=C(C(=O)N1CC=4C=NC=NC4)C32
Molecular Formula
C17H10BrN3O2
Molecular Weight
368.18
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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