LHQ490
Product Specifications
Target
FGFR, Apoptosis
Related Pathways
Angiogenesis, Tyrosine Kinase/Adaptors, Apoptosis
Bioactivity
LHQ490 is a selective FGFR2 inhibitor with an IC50 of 5.2 nM. It effectively suppresses the proliferation of BaF3-FGFR2 cells, with an IC50 value of 1.4 nM. Additionally, LHQ490 inhibits the proliferation of FGFR2-driven cancer cells and induces apoptosis in these cells.
Molecular Formula
C30H33FN6O2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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