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LC-MI-3

Product Specifications

Target

PROTACs, IRAK, NF-κB

Related Pathways

PROTAC, NF-κB, Immunology/Inflammation

Bioactivity

LC-MI-3 is an orally active and potent PROTAC degrader of interleukin-1 receptor-associated kinase 4 (IRAK4), with a DC50 value of 47.3 nM. It effectively inhibits the activation of downstream NF-κB signaling. LC-MI-3 is applicable for research in both acute and chronic inflammatory skin conditions.

Molecular Formula

C39H36N8O8

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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