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AR Degrader-1

Product Specifications

Target

Molecular Glues|||Androgen Receptor|||E1/E2/E3 Enzyme

Related Pathways

Endocrinology/Hormones|||Ubiquitination|||PROTAC

Bioactivity

AR Degrader-1 (Compound ML 2-9) is a monovalent degrader of androgen receptors (AR) categorized under molecular glues. In LNCaP prostate cancer cells, it facilitates AR degradation through DCAF16 (E3 ligase) while exhibiting minimal cytotoxicity.

Molecular Formula

C24H27ClN6O4S

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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