GAT2711
Product Specifications
Target
AChR
Related Pathways
Neuroscience
Bioactivity
GAT2711 is a full agonist of α9nAChR, with an EC50 of 230 nM. It exhibits 340 times greater selectivity for α9 over α7nAChR. In THP-1 cells, GAT2711 inhibits ATP-induced IL-1β release. Additionally, GAT2711 retains full analgesic activity in α7nAChR knockout mice.
Molecular Formula
C20H27IN4O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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