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XYD190

Product Specifications

Target

PROTACs, Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic, PROTAC

Bioactivity

XYD190 (Compound 14g) is an orally active degrader of CBP/p300. It inhibits the bromodomain of CBP/p300 with an IC50 of 483.7 nM and demonstrates antitumor activity against acute myeloid leukemia.

Molecular Formula

C55H50F2N10O7

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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