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4F-DDC

Product Specifications

Target

PARP

Related Pathways

Chromatin/Epigenetic, DNA Damage/DNA Repair

Bioactivity

4F-DDC is a novel PARP1 inhibitor with an IC50 value of 82 nM, which induces DNA damage and activates the cGAS-STING pathway. Additionally, 4F-DDC inhibits the growth of tumors derived from HCC-1937 xenografts.

Molecular Formula

C16H14Br2FN3O2S

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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