Antitumor agent-151
Product Specifications
Target
Apoptosis
Related Pathways
Apoptosis
Bioactivity
Antitumor agent-151 (7k) is a notable HsClpP agonist and a potential candidate for leukemia treatment. This compound significantly boosts the proteolytic activity of HsClpP (EC50= 0.79 μM) and exhibits remarkable in vitro antitumor activity (IC50= 0.038 μM) . Additionally, Antitumor agent-151 (7k) induces apoptosis.
Molecular Formula
C22H20FN5O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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