EGFR kinase inhibitor 6
Product Specifications
Target
Apoptosis, EGFR
Related Pathways
JAK/STAT signaling, Angiogenesis, Tyrosine Kinase/Adaptors, Apoptosis
Bioactivity
EGFR kinase inhibitor 6 (Compound 4b) is an orally active epidermal growth factor receptor (EGFR) kinase inhibitor with an IC50 of 24.34 μM. It induces apoptosis and demonstrates anticancer and anti-inflammatory properties, exhibiting low toxicity with an LD50 range of 500-2000 mg/kg.
Molecular Formula
C21H16ClN3OS2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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