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NZ-97

Product Specifications

Target

Proteasome

Related Pathways

Proteases/Proteasome, Ubiquitination

Bioactivity

NZ-97 is an inhibitor of dipeptidyl peptidase 4 (DPP4) with an IC50 of 18 nM. It exhibits low initial plasma exposure with a Cmax of 0.13 μM and is eliminated within 8 hours. NZ-97 can ameliorate lipopolysaccharides-induced lung injury and bleomycin-induced pulmonary fibrosis in mouse models.

Molecular Formula

C43H67N5O9

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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