PAR4 antagonist 2
Product Specifications
Target
Protease-activated Receptor
Related Pathways
GPCR/G Protein
Bioactivity
PAR4 antagonist 2 (Compound 31) is a protease-activated receptor 4 (PAR4) antagonist with IC50 values of 95 nM for human PAR4 and 367 nM for mouse PAR4. It inhibits the activation of PAR4 through cleavage by the natural protease thrombin but has no effect on the synthetic PAR4 agonist peptide AYPGKF.
Molecular Formula
C22H18F2N6O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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