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Tyrosine kinase-IN-8

Product Specifications

Target

Bcr-Abl

Related Pathways

Cytoskeletal Signaling, Angiogenesis, Tyrosine Kinase/Adaptors

Bioactivity

Tyrosine kinase-IN-8 (compound 4e) is a BCR‐ABL1 tyrosine kinase inhibitor (TKI) exhibiting antiproliferative activity against the chronic myeloid leukemia (CML) cell line K562, with a CC50 of 0.8 μM. Tyrosine kinase-IN-8 is applicable for research in chronic leukemia.

Molecular Formula

C31H21F2N7O2

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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